Pharmacology

Propofol Pharmacology

Propofol (2,6-diisopropylphenol) is the most widely used intravenous induction agent in modern anesthesia practice. Its favorable pharmacokinetic profile — rapid onset, short context-sensitive half-time, and minimal accumulation — makes it suitable for both induction and maintenance of anesthesia. Understanding its hemodynamic effects, dosing adjustments for special populations, and role in total intravenous anesthesia (TIVA) is essential for safe practice.

Key Points

1

GABA-A receptor agonist with rapid onset (30–45 seconds) and short duration (5–10 minutes)

2

Induction dose: 1.5–2.5 mg/kg IV; reduced in elderly and hemodynamically compromised patients

3

TIVA infusion: 100–200 mcg/kg/min maintenance; titrate to clinical effect or BIS 40–60

4

Causes dose-dependent hypotension via decreased SVR and mild myocardial depression

5

Antiemetic properties at sub-hypnotic doses (10–20 mg IV bolus)

Clinical Pearl

In hemodynamically unstable patients, reduce propofol induction dose to 0.5–1 mg/kg and administer slowly over 30–60 seconds. Consider etomidate or ketamine as alternatives when hemodynamic stability is the priority.

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References

[1]Propofol: An Overview of Its Pharmacology.British Journal of Anaesthesia
[2]Propofol Infusion Syndrome: A Structured Review.British Journal of Anaesthesia
[3]TIVA with Propofol: Practical Aspects.Current Opinion in Anaesthesiology

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